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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T23094 | NTNCB hydrochloride | Others , Neuropeptide Y Receptor | |
NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor. | |||
TQ0286 | MK-0557 | Neuropeptide Y Receptor | |
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM). | |||
T10539 | BIBO3304 TFA | Neuropeptide Y Receptor | |
BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 receptor). | |||
T8963 | CYM2503 | Neuropeptide Y Receptor | |
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthosteric galanin binding site of the receptor (as measured by ... | |||
TP2206 | [Leu31,Pro34]-Neuropeptide Y (porcine) | Neuropeptide Y Receptor | |
High affinity neuropeptide Y Y1 receptor agonist | |||
T17222 | Velneperit | S2367 | Neuropeptide Y Receptor |
Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity. | |||
T5455 | HT-2157 | SNAP37889,SNAP-37889 | Neuropeptide Y Receptor |
HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target. | |||
T5587 | CGP71683 hydrochloride | CGP71683A | Neuropeptide Y Receptor |
CGP71683 hydrochloride (CGP71683A) is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM) in cell membranes. | |||
TP1380 | Galanin (1-16), mouse, porcine, rat | Neuropeptide Y Receptor | |
Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons. | |||
T1997 | JNJ-31020028 | JNJ 31020028 | Neuropeptide Y Receptor |
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold selectivity for Y2 versus human Y1/Y4/Y5 receptors. | |||
TP1059 | Peptide YY (PYY) (3-36), human | Peptide YY (3-36) | Neuropeptide Y Receptor |
Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite. | |||
T8456 | GALNON | Neuropeptide Y Receptor | |
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties | |||
T12895 | SHA 68 | Neuropeptide Y Receptor | |
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR)(NPSR Asn107 and NPSR Ile107 with IC50s of 22.0 and 23.8 nM, respectively). | |||
T21611L | BWX 46 Acetate | BWX 46 Acetate(172997-92-1 Free base) | Neuropeptide Y Receptor |
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM. | |||
T23087 | NPY 5RA972 | Neuropeptide Y Receptor | |
neuropeptide Y Y5 receptor antagonist | |||
TP1044L | Pancreatic Polypeptide, rat acetate | Neuropeptide Y Receptor | |
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4. | |||
T24121 | GW438014A | GW 438014 A,GW-438014-A | Neuropeptide Y Receptor |
GW438014A is a potent, selective antagonist of the NPY-Y5 receptor, effectively inhibiting food consumption and curbing body weight gain in obese rodents. | |||
TP1984L | [D-Trp34]-Neuropeptide Y Acetate | [D-Trp34]-Neuropeptide Y Acetate (153549-84-9 Free base) | Neuropeptide Y Receptor |
[D-Trp34]-Neuropeptide Y Acetate is a potent and selective agonist of neuropeptide Y (NPY) Y5 receptor. [D-Trp34]-Neuropeptide acetate Y is a significantly less potent agonist at the NPY Y1, Y2, Y4, and y6 receptors. [D-... | |||
TP1618L | PACAP-38 (31-38), human, mouse, rat acetate | PACAP-38 (31-38), human, mouse, rat acetate(138764-85-9 Free base) | PACAP |
PACAP-38 (31-38), human, mouse, rat acetate is an activator of PAC1 receptor. PACAP-38 (31-38), human, mouse, rat acetate demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY an... | |||
TP1137L | Pancreatic Polypeptide (human) acetate | Neuropeptide Y Receptor | |
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist. |